Proceedings of the  ECHET96 ConferenceNew Synthetic Methodology


Text: Keynote, Stereocontrolled Reactions, New Synthetic Methodology, Reaction Mechanisms and Conformational Analysis and Molecular Modeling and Databases
Graphical Abstracts: Keynote, Stereocontrolled Reactions, New Synthetic Methodology, Reaction Mechanisms and Conformational Analysis and Molecular Modeling and Databases

004John W. Lyga*, Syed F. Ali, Charles A. Webster, Kirk A. Simmons, Marjorie J. Plummer and Malgorzata E. Galietti Synthesis And Evaluation Of An "Indexed" Combinatorial Library For Lead Optimization
Poster Received 01/Apr/1996ECHET96 Contribution 004: Graphical Abstract
016C. Oliver Kappe and Albert Padwa* Furo[3,4-b]indoles and Thieno[2,3-c]furans via a Pummerer Induced Cyclization Reaction
Poster Received 22/Apr/1996ECHET96 Contribution 016: Graphical Abstract
055Hideshi Nakamura, Daisuke Takeuchi, Mihoko Aizawa, Chun Wu and Akio Murai Synthesis of 3,5-disubstituted 2-aminopyrazines by Pd-mediated cross-couplings and its use for preparing chemi- and/or bioluminescent compounds.
Poster Received 26/Apr/1996ECHET96 Contribution 055: Graphical Abstract
074Gordon W. Gribble Erin T. Pelkey Louis Chang David H. Blank A Novel Synthesis of the Pyrrolo[2,3-b]indole Ring System
Poster Received 26/Apr/1996ECHET96 Contribution 074: Graphical Abstract
005Xia Shao, Jeffery Kohrt, Dallas K. Bates Steric Crowding Alters The Reaction Pathway For Sulfoxide Electrophilic Substitution (SES)
Poster Received 03/Apr/1996ECHET96 Contribution 005: Graphical Abstract
006M. Koos, B. Steiner, J. Gajdos Synthesis of Some Bridged Heterocycles with Saccharide Moiety in the Molecule
Poster Received 12/Apr/1996ECHET96 Contribution 006: Graphical Abstract
007Nagatoshi Nishiwaki, Yasuo Tohda, and Masahiro Ariga Nitropyrimidinones: Synthetic Equivalents of Unstable Nitromalonaldehyde and Diformylamine
Poster Received 17/Apr/1996ECHET96 Contribution 007: Graphical Abstract
017Arnaud Tatibouët, Martine Demeunynck, Pierre Vatton, Jean Lhomme Reaction Of 3-Aminoacridine With Formaldehyde In Acidic Media: Access To A Series Of "Fascinating" Molecules
Poster Received 22/Apr/1996ECHET96 Contribution 017: Graphical Abstract
018Vasiliy Bakulev*, Vera Berseneva, Yury Morzherin, Natalia Belskaya, Marina Muhacheva Heterocyclization Of Thioacetamide Derivatives
Poster Received 22/Apr/1996ECHET96 Contribution 018: Graphical Abstract
022Mateo Alajarin and Angel Vidal INTRAMOLECULAR (2+2) CYCLOADDITION IMINE-KETENIMINE
Poster Received 23/Apr/1996ECHET96 Contribution 022: Graphical Abstract
032U. Jordis and B. Küenburg Chiral Bridged Piperazines: Synthesis of (1S,4S) 2,5-Diazabicyclo[2.2.2]octane
Poster Received 24/Apr/1996ECHET96 Contribution 032: Graphical Abstract
036F. Sauter, U. Jordis and P. Martinek Who can model New Quinolone-Type Heterocycles as Potential Antibacterials? Synthesis of Thieno[2',3':4,5]thieno[3,2-b]-pyridone-3-carboxylic acids.
Article Received 24/Apr/1996ECHET96 Contribution 036: Graphical Abstract
042Wolfgang Holzer and Brigitte Plagens Alkylation of Pyrazolones via the Mitsunobu Reaction
Poster Received 25/Apr/1996ECHET96 Contribution 042: Graphical Abstract
043Uno Mäeorg, Ebba Loodmaa Synthesis of (+/-)-3,3,7-trimethyl-2,9-dioxabicyclo[3.3.1.04,7]nonane (lineatin) - the aggregation pheromone of an ambrosia beetle (Trypodendron lineatum)
Poster Received 25/Apr/1996ECHET96 Contribution 043: Graphical Abstract
044Vidar Bjørnstad1, Paul Frøyen1, Håkon Hope2 and Jan Skramstad*1 New Heterocycles from Reaction of Thiomaleic Anhydrides with Trivalent Phosphorus
Article Received 25/Apr/1996ECHET96 Contribution 044: Graphical Abstract
047F. Guillier, F. Nivoliers, A. Godard, F. Marsais and G. Queguiner Metalation connected to Palladium-catalysed cross-coupling strategy: Synthesis of 4,5-disubstituted-benzo[c][2,7]naphthyridines as key intermediates for the synthesis of polycyclic marine alkaloids of pyrido[4,3,2-mn]acridine series.
Article Received 25/Apr/1996ECHET96 Contribution 047: Graphical Abstract
048Karine Couture, Nelly Plé, Alain Turck, Guy Quéguiner* A New Route to Aminodiazines via Metalation Reaction. Synthesis of an Azaanalogue of the Nevirapine.
Poster Received 25/Apr/1996ECHET96 Contribution 048: Graphical Abstract
056Okiko Miyata, Atsuko Nishiguchi, Ichiya Ninomiya, and Takeaki Naito* A Novel Synthesis of Lactones Using Hydroximates as a Tether
Poster Received 26/Apr/1996ECHET96 Contribution 056: Graphical Abstract
057Satoshi MINAKATA, Norio SAKAI, Makoto FUNABASHI, Ilhyong Ryu, Mitsuo KOMATSU Cycloaddition of Novel Mesomeric Betaines, Pyrrolo- and Imidazotriaziniumolates, with Acetylenic Dipolarophiles Leading to Bicyclic Triazocines
Poster Received 26/Apr/1996ECHET96 Contribution 057: Graphical Abstract
059Michael Schoen, Regine Riess, Sabine Laschat, Volker Jaeger 3-Hydroxyisoxazole-5-carbaldehydes - Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles
Poster Received 26/Apr/1996ECHET96 Contribution 059: Graphical Abstract
061Yoshinari Okamoto, Tadashi Okawara, and Mitsuru Furukawa Simple Preparations of Condensed Furan, Perhydropyridazine and Pyrrolidine From Three Components
Poster Received 26/Apr/1996ECHET96 Contribution 061: Graphical Abstract
062Andrea Hajnal, János Wölfling and Gyula Schneider Ring Expansion Of Steroid Oxetans Into Dihydrooxazines
Poster Received 26/Apr/1996ECHET96 Contribution 062: Graphical Abstract
072Ilhyong Ryu, Kazutoshi Matsu, Satoshi Minakata, and Mitsuo Komatsu Novel Synthesis of 2-Pyrrolidinone by Means of Free-Radical Carbonylation
Poster Received 26/Apr/1996ECHET96 Contribution 072: Graphical Abstract
073Mateo Alajarín, Pedro Molina, Pilar Sanchez-Andrada and Concepcion Foces-Foces STUDIES ON CYCLIC CARBODIIMIDES. X-RAY CRYSTAL STRUCTURE OF [a,c]BIS{DIBENZO[d,f][1,3]DIAZEPINO}-1,3-DIAZETIDINE
Poster Received 26/Apr/1996ECHET96 Contribution 073: Graphical Abstract
076R. Alan Aitken and Lawrence Hill CONSTRUCTION OF EXTENDED AND POLYMERIC 1,3-DITHIOLANE AND TETRATHIAFULVALENE DERIVATIVES USING CYCLOADDITION OF Bun3P*CS2
Poster Received 26/Apr/1996ECHET96 Contribution 076: Graphical Abstract
077F. Sauter, J. Fröhlich, S. Chowdhury and C. Hametner Novel One-Pot Double Annelations of Fused Pyrimidine Moieties
Poster Received 26/Apr/1996ECHET96 Contribution 077: Graphical Abstract
081Robert E. Gawley and Silvio Campagna Alkylations of N-allyl-2-lithiopyrrolidines. Several Analogies to Reactions of N-Methyl Compounds, and One Surprise.
Poster Received 26/Apr/1996ECHET96 Contribution 081: Graphical Abstract
083John B. Bremner, Reginald J. Smith and Gregory J. Tarrant. Application of the Meisenheimer Rearrangement to the Synthesis of Hydroxalated Tropane Alkaloid Derivatives
Poster Received 27/Apr/1996ECHET96 Contribution 083: Graphical Abstract
085Reuben Jih-Ru Hwu,* Shwu-Chen Tsay, Zahra Ranezani, and Gholam H. Hakimelahi New bata-Lactam Analogs as Antimicrobial Agents: Design and Synthesis
Poster Received 27/Apr/1996ECHET96 Contribution 085: Graphical Abstract
092Andre chieffia, Victor Snieckusa and Joao V. Comassetob Transmetalation Reaction Of Ferrocenyl Tellurides
Poster Received 27/Apr/1996ECHET96 Contribution 092: Graphical Abstract
001Alexei Nemazany [a] and Norbert Haider [b] Synthesis of Heterocycle-Annelated Naphthyridones with a Bridgehead Nitrogen Atom
Poster Received 01/Apr/1996ECHET96 Contribution 001: Graphical Abstract
010L. Martarello, D. Joseph, D. Prim and G. Kirsch Behavior of 1,3-disubstituted-4,5,6,7-tetrahydrobenzo[c]thiophen-4-one in the Fischer indole synthesis
Poster Received 17/Apr/1996ECHET96 Contribution 010: Graphical Abstract
012Iain Coldham, Alan J. Collis and Roger J. Mould Vinylaziridines from vinylepoxides
Poster Received 18/Apr/1996ECHET96 Contribution 012: Graphical Abstract
019Mario R. Tellez Synthesis of 2-(2-fluorophenylimino-3-(2-fluorophenyl)-1,3-thiazolidine-4,5-dione, di-4-fluorophenyl-thioparabanic acid, and 3-(p-fluorophenyl)-1,3-thiazetidin-4-one-2-(p-fluorophenyl)-imine. Easy and versatile conversion of the thiazetidinone into carbodiimide or isourea derivatives.
Poster Received 22/Apr/1996ECHET96 Contribution 019: Graphical Abstract
024Manuel Garrido, Rosa Dominguez, Ana Martínez, Jacobo Cruces, Elena Martinez, Juan C. Estévez and Ramón J. Estévez. A NEW STRATEGY FOR THE SYNTHESIS OF INDOLONAPHTHOQUINONES AND BENZOFURANONAPHTHOQUINONES.
Poster Received 23/Apr/1996ECHET96 Contribution 024: Graphical Abstract
035F. Sauter, U. Jordis and P. Martinek [1]Benzothieno[3,2-b]pyridone-3-carboxylic Acids as Potential Antibacterials
Article Received 24/Apr/1996ECHET96 Contribution 035: Graphical Abstract
046Patricia CHARPENTIER, Jean-François BRIERE, Georges DUPAS,

Guy QUEGUINER and Jean BOURGUIGNON

Design And Synthesis Of A Heterocyclic Amine Receptor
Poster Received 25/Apr/1996ECHET96 Contribution 046: Graphical Abstract
052Akikazu Kakehi, Suketaka Ito, and Fumihito Ishida Synthesis and Rearrangement of 5aH-Pyrido[1,2-d][1,3,4]thiadiazepine Derivatives
Poster Received 26/Apr/1996ECHET96 Contribution 052: Graphical Abstract
066Takeo Konakahara, Yoshitomo Ono, and Sanae Tamura Reaction of a-trimethylsilylmethyl-substituted aromatic N-heterocycles with methyl perfluoro(2-methyl-1-propenyl) ether
Poster Received 26/Apr/1996ECHET96 Contribution 066: Graphical Abstract
097F. Sauter, J. Fröhlich and M. Pfalz Syntheses of Novel 3-Hetero-spiro[5,5]-undecane-9-ones and Reactions Thereof
Poster Received 29/Apr/1996ECHET96 Contribution 097: Graphical Abstract
103M. A. Kuznetsov, L. M. Kuznetsova, J. G. Schantl Azimines, Azo-aziridines, 1,2,3-Triazoles. Products obtained from the Oxidation of N-aminophthalimide in the presence of Azo-alkenes.
Poster Received 30/Apr/1996ECHET96 Contribution 103: Graphical Abstract
104E.V.K. Suresh Kumar*, J.D. Singh and H.B. Singh A Convenient Synthesis Of 5-Methylthieno[2,3-D]-1,3-Dithiole-2-Thione And Its Tetrathiafulvalene (TTF)
Poster Received 30/Apr/1996ECHET96 Contribution 104: Graphical Abstract
115Stefano C.G. Biagini, Vernon C. Gibson, Edward L. Marshall, Michael North,a and Paul Williams The Synthesis and ROMP of Heterocyclic Monomers
Poster Received 03/Jun/1996ECHET96 Contribution 115: Graphical Abstract
117Fernando Cortes G., Gustavo Avila Z. and Lius Angel Maldonado G. A simple modification to improve the generality of Terry's 3,4-dusubstituted pyrrole synthesis
Poster Received 11/Jun/1996ECHET96 Contribution 117: Graphical Abstract
118Reyna Diaz-Cortes F., Ana L. Silva P. and Luis Angel Maldonado G. A simple approach to 2-substituted 4-furanemethanol compounds
Poster Received 11/Jun/1996ECHET96 Contribution 118: Graphical Abstract
120Ganesh Pandey* and M. Karthikeyan Novel Construction of Benzazocine Framework through Photoinduced Electron Transfer (PET) Generated Arene Radical Cation.
Poster Received 23/Apr/1996ECHET96 Contribution 120: Graphical Abstract

Text: Keynote, Stereocontrolled Reactions, New Synthetic Methodology, Reaction Mechanisms and Conformational Analysis and Molecular Modeling and Databases
Graphical Abstracts: Keynote, Stereocontrolled Reactions, New Synthetic Methodology, Reaction Mechanisms and Conformational Analysis and Molecular Modeling and Databases

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