Synthesis and evaluation of an "indexed" combinatorial library for lead optimization

Footnotes

  1. Krapcho, J, Turck, C. F, U.S. Patent No. 4,065,617 (Dec. 27, 1977), 3,931,169 (Jan. 6, 1976), 3,923,816 (Dec. 2, 1975), 3,911,129 (Oct. 7, 1975) all assigned to E. R. Squibb.
  2. Krapcho, J, Turck, C. F, U.S. Patent No. 3,926,968 (Dec. 16, 1975) assigned to E. R. Squibb.
  3. Pirrung, M. C., Chen, J., J. Am. Chem. Soc., 1995, 117, 1240.
  4. Smith, P. W., Lai, J. Y. Q., Whittington, A. R., Cox, B., Houston, J. G., Stylli, C. H., Banks, M. N., Tiller, P. R., Bioorg. Med. Chem. Let., 1994, 4, 2821.

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